常用名 盐酸替扎尼定

英文名 Tizanidine hydrochloride

CAS号 64461-82-1

沸点 391.2ºC at 760 mmHg

熔点 280 °C

分子式 C9H9Cl2N5S

分子量 290.17200

闪点 190.4ºC

精确质量 288.99600

PSA 90.44000

LogP 2.35520

外观性状 白色固体

储存条件 存放在密封容器内，并放在阴凉，干燥处。储存的地方必须远离氧化剂，远离热存放。

稳定性 远离氧化物，热，光。

水溶解性 H2O: ~29 mg/mL

"Tizanidine hydrochloride is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.

Target: α2-adrenergic receptor

Tizanidine is a drug that is used as a muscle relaxant. It is a centrally acting α2 adrenergic agonist. It is used to treat the spasms, cramping, and tightness of muscles caused by medical problems such as multiple sclerosis, ALS, spastic diplegia, back pain, or certain other injuries to the spine or central nervous system. It is also prescribed off-label for migraine headaches, as a sleep aid, and as an anticonvulsant. It is also prescribed for some symptoms of fibromyalgia.

Tizanidine has been found to be as effective as other antispasmodic drugs and has superior tolerability to that of baclofen and diazepam. Tizanidine can be very strong even at the 2 mg dose and may cause hypotension, so caution is advised when it is used in patients who have a history of orthostatic hypotension, or when switching from gel cap to tablet form and vice versa. Tizanidine can occasionally cause liver damage, generally the hepatocellular type. Clinical trials show that up to 5% of patients treated with tizanidine had elevated liver function test values, though symptoms disappeared upon withdrawal of the drug. Care should be used when first beginning treatment with tizanidine with regular liver tests for the first 6 months of treatment."

包装：100mg，500mg，1g，10g，100g以及kg级别等公斤级大包装

纯度：99%

配送：惯例下常温**

包装：袋装

厂家：西安齐岳生物科技有限公司

关于我们：

西安齐岳生物科技有限公司具备批量生产能力和强大的研发能力，这样的双重优势可以确保企业不仅在满足市场需求上保持高效，同时也在产品创新和技术升级。能够提供100mg，500mg，1g，10g，100g以及kg级别等公斤级大包装。

相关产品：

CAS:20123-80-2 Calcium dobesilate

CAS:53251-94-8 Pinaverium bromide

CAS:2870-71-5 Atropine methyl (bromide)