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CAS: 3031330-66-9 ML 2-23PROTAC Hemagglutinin Degrader-1 PROTACs(蛋白降解靶向嵌合体)
发布时间:2024-04-23     作者:kx   分享到:

常用名:PROTAC Hemagglutinin Degrader-1 

描述:

PROTAC Hemagglutinin Degrader-1 (Compound V3) 是一种有效的 PROTAC 流感病毒血凝素 (influenza hemagglutinin (HA)) 降解剂,降解中值浓度为 1.44 μM。

生物活性

PROTAC Hemagglutinin Degrader-1 (Compound V3) is a potent PROTAC influenza hemagglutinin (HA) degrader with a median degradation concentration of 1.44 μM. PROTAC Hemagglutinin Degrader-1 shows broad-spectrum anti-influenza virus activity[1].


体内研究

(In Vivo)

PROTAC Hemagglutinin Degrader-1 (0-20 mg/kg; i.v.; daily for 5 days) protects mice against influenza A virus-induced toxic effects[1].

PROTAC Hemagglutinin Degrader-1 displays a moderate oral bioavailability of approximately 6.8%[1].


MCE has not independently confirmed the accuracy of these methods. They are for reference only.


分子量 1072.48


Formula C61H93N5O9S


CAS 号 3031330-66-9


运输条件 Room temperature in continental US; may vary elsewhere.


储存方式 Please store the product under the recommended conditions in the Certificate of Analysis.

CAS:	3031330-66-9	ML 2-23PROTAC Hemagglutinin Degrader-1     PROTACs(蛋白降解靶向嵌合体)

产地:西安

用途:科研

厂家:西安齐岳生物科技有限公司

温馨提示:仅用于科研!

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